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プロポフォール - アストラゼネカ AstraZeneca
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1. 8 4 738 1 369 28 9 364 11 9 414 8 7 161 3 4 1 F 1 2 3 4 5 6 8 9 10
2. i 12 0 02SmL kg 10 Ni 1 2 1
3. 0 1 0 13 0 1 0 1 0 15 0 1 CK CPK
4. 0 1 0 1 0 1 5 0 1 gt 5 0 15 0 15 0 1
5. 10 1 20 2 12 6 SD 11 Cs
6. a 95 x g mL 0 T T T T 2 3 4 5 6 mg kg 0 727 X 0 238 Richards 95 3 116 99 1 113 116 0 3 3 0mg kg 100 25 25 21 10 8 3 12 7 8 121 4 3 3 6 AST GOT ALP LDH
7. TCI TCI
8. AUCo 8 2 6mg kg 24 1 4 1 4 68 3 9 10 120 7 97 99 2 5mg kg 8 V CLrg 20 25
9. 1 2 3 4 5 TCTI
10. 3 0uug mL 2 0 5 0ug mL G 102 0gmL 1 2 1 7 PR 7 0 5 3 ES 0 03 0 30mL kg 003mKke 1 ASAT IV 1 2 0 025mL kg 10
11. 4 5 Propofol JAN 2 6 Diisopropylphenol OH 0 HC CH Ne Hs C CH CHiaO 178 27 99 5 2 3 MRI TCTI
12. 0 03mL kg 0 3mg kg 3 Ramsay score 3 0 03 0 3mL kg 0 3 3 0mgkg 1 30 HDso 12 9mg kg 50 LDs 57 9mg kg LDHDs 4 2 HDs 2 3 3
13. 1 TCI 1 0 05SmL kg 10 0 Smg kg 10 1 2 3 0 20 0 2SmL kg 2 0 2 5mg kg 2 30 100 10 1 0mL kg 10mg kg 10 0 8mL kg 8mg kg 0 6mL kg 6mgkg 0 4 1 0mL kg
14. lt 3 da 4 I 5 1 2 3 1 1 1
15. 11 0 1 2 5 0 1 5 0 1 ST AST GOT ALT GPT Al P LDH 7 GTP
16. SS TY Bg 1 62 2 TCI 1 10 gt 20 20 gt 30 3 gt 1 0mL kg 0 8mL kg 0 6mL kg 10mgkg 8mg kg 6mgkg TCTI NR TCT WW i
17. 2 TCI TOT 3 3 1 1 2
18. 3 4 G 5 5 2mg mL MM lt 6 DEHP di 2 ethylhexyD phthalate 2 DEHP
19. 1 TCI 3 3 6 3L CLrs 7 202D 1 TCI 1 2 3 709 0 Smg kg 10 100 709 709 2 21 0 39mg kg 46 99 2 124 125
20. 0 4 1 0mL kg OO Omg kg 5 775 Co a 5 2 TCI 1 A t 3 04ug mL 3 ER ER 1 1 0 2 0ug mL ji AT Em yx HL 0 3 0 6 0ug mL 1 3 a 1 1 mL kg ASATI IV mg kg
21. I 2 es 0 03mL kg NE 8 0 3mg kg 1 TCTI I NT i NE 2 TCI 0 03 0 30mL kg 0 3 3 0mg kg 3 TCI i TCI AA A TCT
22. TCI 5 100 55 55 3 15ug mL 1 8 2 80g mL 11 4 1 08 1 91gmL 1 53 33 60 0 38 49 1 9 1 7 3 1 8 7 GTP 1 8 wg m 10 68 r 0 809 T T T 1 gg mL 9 10 1 3 y x 70kg 120
23. lt
24. 4 1200mL 10 es 2 4 gmD 1300 1200 F1100 1000 7 600 3 F900 6d 800 F700 9 LT 0 0 600 PB 0 2 _ om F300 KN 3 F400 2 F300 F200 1 Li00 0 1 T 0 0 10 20 30 40 50 60 70kg 40 10 3ug mL 10 2 g mL 10 3ug mL 30 TCI 4 4
25. 4 10mg kg 2 TCI 3 0 g mL 1 2 3 3 1 1 0 2 0g mL 3 0 6 0g mL 2 0 5 0g mL TCI
26. TCI 1 0 05mL kg 10 0 5mgkg 10 MFJ ASAT TV 1 7 25 3 0 20 0 25mL kg a TA TY 2 0 2 5mg kg Gm me 100mg 1 22 5mg 2 a 1mL 12 EE 0 035mg pH 2 196
27. TCTI a 19 20mL 1 50mL 1 1 Bennett S N et al New Eng J Med 333 3 147 1995 2 Parke T J et al Br Med J 305 6854 613 1992 3 39 219 683 1990 4 Kay NH et al Br J Anaesth 38 1075 1986 5 29 1 77 1993 6 Kirkpatrick T et al Br J Anaesth 60 146 1988 7 Dyck B J et al Semin Anesth 11 2 1992 8 Swinhoe C F et al Anaesthesia 53 Suppl 1 61 1998 1 9 Morcos W E et al Posterad Med J 61 Suppl 3 62 1985 3 CE i 10 Ickx B et al Br J Anaesth 81 854 1998 0 11 Servin F et al Anesthesiology 69 887 1988 Servi
28. 2 4 5 1 0mL 0 1g 7 1 lt 2
29. Brugada V1 V3 coved ST 5 3 1 9 3 0 tiz8 365 tiz7 51 6 1 0 2 0 2 5mg kg 2 6 ti a 3 26L 317L CLrs 1 62L 1C 2 5mg kg
30. 433 99 8 432 433 4 10mg kg 7 6 97 2 69 71 1 167 240 20 6 269 12 4 5 1 1 3 0 9 0 7 0 5 1 167 60 1 AST GOT ALT GPT LDH 7 GTP 38 12 31 6 13 28 9 2 TCI
31. PE II gmL 2 TCI Target Controlled mfusion TCI TCI oe 2 0 5 0g mL 2 1 TCI 3 a 13 TC 9 1
32. TCI 100 90 80 TCI F 60 50 40 30 TCI L 50 T T T T T T T 0 0 15 30 45 60 75 90 105 120 2 4 I 3 15 g mL 3 2 80gmL TCT 2 08mgkg 40 1 5 8sSmg kg 2 54 10 Raftery 61 5 10 7 6 4mg kg 3 3 6 4 5 3 6 3 2 4mg kg 3 TCI
33. 4 12 12 6 1 3 2 TCTI TCI
34. J et al Br J Anaesth 65 157 1990 26 32 2 95 1996 27 32 2 105 1996 _ a 28 Glen J B Br J Anaesth 52 731 1980 29 Tomoda K et al Br J Anaesth 71 383 1993 330 0011 3 1 0120 189 115 FAX 06 6433 7376 AstraZeneca 1995 AstraZeneca 3 1 DPFS PI710 CH51M
35. DPFS 9 0 2013 1 13 2012 12 871119 21300AMY00077 rl 8 20orfel 2001 6 lz 23 2 a Diprivan Injectionskit 1 1
36. n F et al Br J Anaesth 65 177 1990 a Barvais L et al J Cardiothorac Vasc Anesth 10 7 877 1996 Servin F et al Anesthesiology 78 657 1993 29 1 3 1993 29 1 11 1993 34 2 109 1998 34 2 121 1998 23 TCI 2001 24 Raftery S et al Br J Anaesth 66 566 1991 NN NY DD CO O DD 01 29 1 23 1993 29 1 33 1993 29 1 45 1993 29 1 57 1993 25 Richards M
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